Search results for "Anti proliferative"

showing 2 items of 2 documents

Experimental and theoretical study of possible correlation between the electrochemistry of canthin-6-one and the anti-proliferative activity against …

2015

Abstract This work presents an approach to study the performance of novel targets able to overcome cancer stem cell chemoresistance, based on the voltammetric data for microparticulate films of natural or synthetic alkaloids from the canthin-6-one series. A comparison of this voltammetric technique with conventional solution phase electrochemistry suggests the differences in the anti-proliferative activity of canthin-6-ones could be tentatively correlated to their different capacity to generate semiquinone radical anions. These data also match theoretical calculations.

SemiquinoneMolecular modelStereochemistryChemistryOrganic ChemistryAnti proliferativeElectrochemistryCombinatorial chemistryAnalytical ChemistryInorganic ChemistryCancer stem cellCanthin-6-oneStem cellSpectroscopyHuman cancerJournal of Molecular Structure
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Daphne striata Tratt. and D. mezereum L.: a study of anti-proliferative activity towards human cancer cells and antioxidant properties

2018

In this study, we investigated for the first time the anti-proliferative and antioxidant properties of D. mezereum and D. striata. The aerial parts were extracted by maceration with n-hexane, dichloromethane, and methanol. MPLC, GC, and GC-MS were used for the phytochemical study. The anti-proliferative activity was tested against MCF-7, A549, LNCaP, ACHN, and C32 cancer human cells. The antioxidant activity was measured by employing β-carotene bleaching, ABTS, DPPH, and FRAP tests. The Relative Antioxidant Capacity Index (RACI) was applied from the perspective of statistics. D. mezereum dichloromethane extract showed a remarkable anti-proliferative with an IC50 of 6.08 μg/mL against LNCaP …

antiproliferative activityAntioxidantmedicine.medical_treatmentantioxidant activityPlant ScienceDaphne mezereumD. striata01 natural sciencesBiochemistryDaphne mezereum; D. striata; Thymelaeaceae; antiproliferative activity; human tumour cells; antioxidant activityAnalytical ChemistryMaceration (wine)medicinebiologyDaphne striataTraditional medicine010405 organic chemistryfungiOrganic ChemistryAnti proliferativebiology.organism_classification0104 chemical sciences010404 medicinal & biomolecular chemistryDaphne mezereumThymelaeaceaeThymelaeaceaehuman tumour cellsHuman cancer
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